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N/A N=21 Other

Buprenorphine Disposition and CYP3A

Healthy

Enrolled (actual)
21
Serious AEs
0.0%
Results posted
Jan 2020
Primary outcome: Primary: Plasma Cmax of Buprenorphine

Study Design & Population

Study type
Interventional
Phase
N/A
Interventions
Buprenorphine Control (Drug); Buprenorphine + Rifampin (Drug); Buprenorphine + Grapefruit juice (Drug); Buprenorphine + Ketoconazole (Drug)
Age
Adult · 18+ yrs
Sex
All
Sponsor
Washington University School of Medicine
Primary completion
Mar 2014

Outcome Measures

OutcomeResultp-value
PRIMARY
Plasma Cmax of Buprenorphine

Summary

To evaluate role of CYP3A in buprenorphine disposition and effect

Eligibility Criteria

Inclusion Criteria

Each subject must meet all of the following criteria:

  • Male or non-pregnant female volunteer, 18-50 yr old
  • Good general health with no known major medical conditions
  • BMI < 33
  • Provide informed consent

Exclusion Criteria

Subjects will not be enrolled if any of the following criteria exist:

  • Known history of liver or kidney disease
  • Use of prescription or non-prescription medications, herbals or foods known to be metabolized by or affect CYP3A activity (this includes the use of oral contraceptives).
  • Females who are pregnant or nursing
  • Known history of drug or alcohol addiction (prior or present addiction or addiction treatment)
  • Direct physical access to and routine handling of addicting drugs in the regular course of duty (this is a routine exclusion from studies of drugs with addiction potential)
View full record on ClinicalTrials.gov →

Data sourced from ClinicalTrials.gov (NCT01576575). Outcome figures and adverse-event rates are extracted automatically from the registry's posted results and are provided for clinician reference, not as a substitute for the primary publication.

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