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Phase 3 N=19 Treatment

Long Term, Follow-on Study of Lomitapide in Patients With Homozygous Familial Hypercholesterolemia

Familial Hypercholesterolemia

Enrolled (actual)
19
Serious AEs
36.8%
Results posted
May 2018
Primary outcome: Primary: Percent Change in Low Density Lipoprotein Cholesterol (LDL-C) — -45.5 Percent Change

Study Design & Population

Study type
Interventional
Phase
Phase 3
Interventions
lomitapide (Drug)
Age
Adult, Older Adult · 18+ yrs
Sex
All
Sponsor
Aegerion Pharmaceuticals, Inc.
Primary completion
Sep 2012

Outcome Measures

OutcomeResultp-value
PRIMARY
Percent Change in Low Density Lipoprotein Cholesterol (LDL-C)
-51.1
SECONDARY
Percent Change in Low Density Lipoprotein Cholesterol (LDL-C)
-51.1
SECONDARY
Percent Change in Low Density Lipoprotein Cholesterol (LDL-C)
-51.1
SECONDARY
Percent Change in Low Density Lipoprotein Cholesterol (LDL-C)
-51.1
SECONDARY
Percent Change in Low Density Lipoprotein Cholesterol (LDL-C)
-51.1
SECONDARY
Percent Change in Low Density Lipoprotein Cholesterol (LDL-C)
-51.1
SECONDARY
Percent Change in Total Cholesterol
-43.9
SECONDARY
Percent Change in Total Cholesterol
-43.9
SECONDARY
Percent Change in Total Cholesterol
-43.9
SECONDARY
Percent Change in Total Cholesterol
-43.9
SECONDARY
Percent Change in Total Cholesterol
-43.9
SECONDARY
Percent Change in Total Cholesterol
-43.9
SECONDARY
Percent Change in Apolipoprotein B (Apo B)
-60.9
SECONDARY
Percent Change in Apolipoprotein B (Apo B)
-60.9
SECONDARY
Percent Change in Apolipoprotein B (Apo B)
-60.9
SECONDARY
Percent Change in Apolipoprotein B (Apo B)
-60.9
SECONDARY
Percent Change in Apolipoprotein B (Apo B)
-60.9
SECONDARY
Percent Change in Apolipoprotein B (Apo B)
-60.9
SECONDARY
Percent Change in Triglycerides
29.2
SECONDARY
Percent Change in Triglycerides
29.2
SECONDARY
Percent Change in Triglycerides
29.2
SECONDARY
Percent Change in Triglycerides
29.2
SECONDARY
Percent Change in Triglycerides
29.2
SECONDARY
Percent Change in Triglycerides
29.2
SECONDARY
Percent Change in Non High Density Lipoprotein Cholesterol (Non-HDL-C)
-46.6
SECONDARY
Percent Change in Non High Density Lipoprotein Cholesterol (Non-HDL-C)
-46.6
SECONDARY
Percent Change in Non High Density Lipoprotein Cholesterol (Non-HDL-C)
-46.6
SECONDARY
Percent Change in Non High Density Lipoprotein Cholesterol (Non-HDL-C)
-46.6
SECONDARY
Percent Change in Non High Density Lipoprotein Cholesterol (Non-HDL-C)
-46.6
SECONDARY
Percent Change in Non High Density Lipoprotein Cholesterol (Non-HDL-C)
-46.6
SECONDARY
Percent Change in Very Low Density Lipoprotein Cholesterol (VLDL-C)
30.6
SECONDARY
Percent Change in Very Low Density Lipoprotein Cholesterol (VLDL-C)
30.6
SECONDARY
Percent Change in Very Low Density Lipoprotein Cholesterol (VLDL-C)
30.6
SECONDARY
Percent Change in Very Low Density Lipoprotein Cholesterol (VLDL-C)
30.6
SECONDARY
Percent Change in Very Low Density Lipoprotein Cholesterol (VLDL-C)
30.6
SECONDARY
Percent Change in Very Low Density Lipoprotein Cholesterol (VLDL-C)
30.6
SECONDARY
Percent Change in Lp(a)
-10.4
SECONDARY
Percent Change in Lp(a)
-10.4
SECONDARY
Percent Change in Lp(a)
-10.4
SECONDARY
Percent Change in Lp(a)
-10.4
SECONDARY
Percent Change in Lp(a)
-10.4
SECONDARY
Percent Change in Lp(a)
-10.4
SECONDARY
Percent Change in High Density Lipoprotein Cholesterol (HDL-C)
-23.5
SECONDARY
Percent Change in High Density Lipoprotein Cholesterol (HDL-C)
-23.5
SECONDARY
Percent Change in High Density Lipoprotein Cholesterol (HDL-C)
-23.5
SECONDARY
Percent Change in High Density Lipoprotein Cholesterol (HDL-C)
-23.5
SECONDARY
Percent Change in High Density Lipoprotein Cholesterol (HDL-C)
-23.5
SECONDARY
Percent Change in High Density Lipoprotein Cholesterol (HDL-C)
-23.5
SECONDARY
Percent Change in Apolipoprotein AI (Apo AI)
-30.5
SECONDARY
Percent Change in Apolipoprotein AI (Apo AI)
-30.5
SECONDARY
Percent Change in Apolipoprotein AI (Apo AI)
-30.5
SECONDARY
Percent Change in Apolipoprotein AI (Apo AI)
-30.5
SECONDARY
Percent Change in Apolipoprotein AI (Apo AI)
-30.5
SECONDARY
Percent Change in Apolipoprotein AI (Apo AI)
-30.5

Summary

This was a long term follow on study to assess the continued long term safety and efficacy of lomitapide in patients with homozygous familial hypercholesterolemia.

Eligibility Criteria

Inclusion Criteria

  • Completed UP1002 or 733-005.
  • Willing and able to provide consent and comply with the requirements of the study protocol.

Exclusion Criteria

  • Met any of the stopping rules for study discontinuation at the final visit of study UP1002 or 733-005.
View full record on ClinicalTrials.gov →

Data sourced from ClinicalTrials.gov (NCT00943306). Outcome figures and adverse-event rates are extracted automatically from the registry's posted results and are provided for clinician reference, not as a substitute for the primary publication.

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